Triptorelin 2mg (10 Vials / Kit)

Triptorelin at a glance

Triptorelin is a decapeptide analog of gonadotropin-releasing hormone, the hypothalamic signal that controls pituitary release of LH and FSH. Replacing the glycine at position six with D-tryptophan makes the molecule far more resistant to enzymatic breakdown and increases its receptor affinity compared with the natural hormone, while the C-terminal glycinamide is retained. In approved medicines it is formulated as acetate or pamoate salts, including sustained-release preparations.

Price and availability

This is SSRBIO‘s kit of 10 vials at 2mg each (20 mg in total), dispatched from China. $67.50 buys the whole kit, which is $3.38/mg. 2 brands currently sell Triptorelin here, so compare their listings before ordering. As with every order here, the brand is paid only after you confirm delivery.

What it is studied for

Triptorelin binds the GnRH receptor on pituitary gonadotroph cells. Initial binding stimulates a surge in LH and FSH release, often called the flare effect, along with a temporary rise in testosterone or estradiol. With sustained receptor occupancy, gonadotrophs become desensitized and receptor numbers fall, so LH and FSH output drops and gonadal sex-steroid production is suppressed to very low levels. That paradoxical outcome, stimulation turning into suppression, is the basis for its clinical use and for research models of reversible hormonal suppression.

Research and regulatory status

Triptorelin is an established prescription medicine, approved in the US, Europe and elsewhere for advanced prostate cancer, and in various regions for endometriosis, uterine fibroids, central precocious puberty and as part of assisted-reproduction protocols. Its clinical pharmacology is documented in decades of trials. Research use covers reproductive endocrinology and hormone-dependent cancer models. Research-grade powder is not an approved formulation and is unrelated to those products' regulatory approvals.

Checking the lab data

A credible report should confirm identity by mass spectrometry matching the calculated mass of the triptorelin decapeptide, and state the salt form, usually acetate, since counter-ions affect weight-based content. HPLC purity should come from a lot-specific chromatogram, and chiral analysis confirming the D-tryptophan configuration adds confidence, because an L-isomer impurity would have the same mass. The lyophilized cake should be white.

No independent report is attached to this listing yet. You can compare brands that publish one on the marketplace or browse the lab reports directory.

Listing details

Compound

Triptorelin

Vial strength

2mg

Vials per kit

10

Total content

20 mg

Price per mg

$3.38

Sold by

SSRBIO

Ships from

China

Lab report

Not yet published

Storage and preparation

Keep unopened freeze-dried vials cold, sealed and out of the light; moisture is what degrades a lyophilized cake fastest. After reconstitution, refrigerate the solution and work within the stability window your protocol sets.

Concentration arithmetic: one 2 mg vial dissolved in 2 mL gives 1 mg/mL, or 2 mg/mL in 1 mL. The Research Lab calculator in your dashboard handles any other volume.

Buyer questions

Supplied for laboratory research only. Not for human or veterinary use, and not a substitute for any prescription medicine. Nothing on this page is medical advice.